- 作者: 蔡明睿、孫珮珮、張夢楊、張彥誠
- 作者服務機構: Department of Chemistry, National Sun Yat-Sen University, Kaohsiung 804, Taiwan, R.O.C.
- 中文摘要: A new route towards the synthesis of N-substituted-4-formylpiperidine using N-benzyl or tryptaminylsulfonylacetamide and a,b-unsaturated ester as starting materials is described. Formal synthesis of AriceptR, deethylibophyllidine, and isoguvacine, which have potential biological activities, were synthesized via this strategy.
- 英文摘要: --
- 中文關鍵字: Stepwise [3+3] annulation; Alane reduction; Dehydrosulfonated; N-substituted-4-formyl piperidine.
- 英文關鍵字: --