- 作者: 吳吉輝; 江彰吉; 黃雅勇; 楊寶旺
- 作者服務機構: Department of Chemistry, Chung Yuan Christian University, Chung-Li, Taiwan 320
- 中文摘要: The Friedel-Crafts reaction of 1-azaazulan-2-ones with .alpha.-haloacid chloride in the presence of aluminum trichloride gives the corresponding .alpha.-haloacyl derivatives. Treatment of these reaction products first with various secondary amines and then with sodium borohydride gives new adrenergic active amine derivatives.
- 英文摘要: --
- 中文關鍵字: Friedel-Crafts reaction; Nucleophilic Substitution; 3-(.alpha.-haloacyl)-1-azaazulan-2-ones; 3-(.alpha.-aminoacyl)-1-azaazulan-2-ones; sodium borohydride; 1-(1-azaazulan-2-onyl-3)-aminoalcohols.
- 英文關鍵字: Friedel-Crafts reaction; Nucleophilic Substitution; 3-(.alpha.-haloacyl)-1-azaazulan-2-ones; 3-(.alpha.-aminoacyl)-1-azaazulan-2-ones; sodium borohydride; 1-(1-azaazulan-2-onyl-3)-aminoalcohols.